产品简要
公司名称 :
Tocris Bioscience
产品类型 :
化学品
产品名称 :
CGP 55845 hydrochloride
目录 :
1248/10
规格 :
10 mg (also 50 mg)
价格 :
269美元
更多信息或购买 :
文章摘录数: 105
参考文献
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产品信息
品牌 :
Tocris, a Bio-Techne Brand
catalog number base :
1248
SKU号 :
1248/10
产品名称 :
CGP 55845 hydrochloride
描述 :
Potent and selective GABAB antagonist
靶标 :
GABA-B Receptor Antagonists
类别 :
Small Molecules
单位尺寸 :
10 mg (also 50 mg)
纯度 :
98%
观察到的分子量 :
438.71
网址印刷 :
?utm_source=labome&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
功能细节 :
CGP 55845 hydrochloride is a potent, selective GABAB receptor antagonist (IC50 = 5 nM) that prevents agonist binding (pKi = 8.35) and inhibits GABA and glutamate release (pEC50 values are 8.08 and 7.85 respectively). Inhibits GABAB responses to baclofen (IC50 = 130 nM in an isoproterenol assay) and potentiates the hypoglycemic response to glucose in vitro .
extended description :
Potent and selective GABAB antagonist
化学品名文本 :
(2S)-3-[[(1S)-1-(3,4-Dichlorophenyl)ethyl]amino-2-hydroxypropyl](phenylmethyl)phosphinic acid hydrochloride
配方 :
C 18 H 22 Cl 2 NO 3 P.HCl
配方文本 :
C18H22Cl2NO3P.氯化氢
cas num :
149184-22-5
美元 :
269美元
产品细节 :
Potent and selective GABAB antagonist
储存 :
存放在RT
更多信息或购买 :
公司信息
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
公司总部: 英国