产品简要
公司名称 :
Tocris Bioscience
产品类型 :
化学品
产品名称 :
毫克132
目录 :
1748/5
规格 :
5毫克
价格 :
166美元
更多信息或购买 :
文章摘录数: 60
参考文献
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产品信息
品牌 :
Tocris
MasterCode :
1748
SKU号 :
1748/5
产品名称 :
毫克132
靶标 :
Calpain Inhibitors
类别 :
Small Molecules
单位尺寸 :
5毫克
纯度 :
95%
观察到的分子量 :
475.63
网址印刷 :
?utm_source=biocompare&utm_medium=referral&utm_campaign=product&utm_term=smallmolecules
功能细节 :
MG 132 is a potent cell-permeable inhibitor of proteasome (IC50 = 100 nM) and calpain (IC50 = 1.2 M). MG 132 inhibits TNF- -induced NF- B activation and I B degradation. Induces neurite outgrowth in PC12 cells and has anticancer properties in vitro . MG 132 inhibits SARS-CoV-2 Mpro in vitro (IC50 = 3.9 M) and inhibits viral replication. Also enhances adeno-associated viral transduction efficiency of human cell lines by around 50-fold.
extended description :
Proteasome and calpain inhibitor. Inhibits NF- B activation
化学品名文本 :
N-[(Phenylmethoxy)carbonyl]-L-leucyl-N-[(1S)-1-formyl-3-methylbutyl]-L-leucinamide
配方 :
C 26 H 41 N 3 O 5
配方文本 :
C26H41N3O5
cas num :
133407-82-6
美元 :
166美元
产品细节 :
Proteasome and calpain inhibitor. Inhibits NF- B activation
别名 :
Z-LLL-al, Z-Leu-Leu-Leu-CHO
储存 :
存放在-20°C
更多信息或购买 :
公司信息
Tocris Bioscience
The Watkins Building
Atlantic Road
Avonmouth, Bristol
BS11 9QD
info@bio-techne.com
https://www.tocris.com
800-343-7475
公司总部: 英国